Posts Tagged ‘antiestrogen’

If you have been hesitating to join the “rewarding” world of anabolic steroids and performance enhancing drugs due to the associated side effects such as excess estrogen formation then Arimidex is one antiestrogen that you can trust easily.

Arimidex, also known as Anastrozole, is an antiestrogen admired by sportsmen on steroids for preventing bloating, oily skin, gynecomastia, acne, and fluid retention. It is worthwhile to note here that these side effects are commonly associated with use of harsh and aromatizable steroids besides androgens and derivatives of testosterone.

The drug is approved by the FDA for treating breast cancer in post-menopausal women with disease progression after the standard therapy, Tamoxifen, has failed to deliver expected results.

The chemical name of Arimidex is 2-[3-(1-cyano-1-methyl-ethyl)- 5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]- 2-methyl- propanenitrile and its has the molecular formula of C₁₇H₁₉N₅. Arimidex has the molecular weight of 293.366 g/mol at the base.

The recommended dose of Arimidex is 0.25-1.0 mg per day or 0.5-1.0 every other day. This drug is best taken with Finasteride because while Arimidex can take care of estrogen production, Finasteride can take care of conversion of Testosterone to DHT (dihydrotestosterone).

When abused, Arimidex can lead to side effects such as shortness of breath, dizziness, diarrhea, vomiting, headache, hat flashes, weakness, cough, and dry mouth. In case of an overdose, it is recommended to contact your nearest medical center. The drug is not indicated to people having an existing allergy to Arimidex or any of its ingredients and is also not recommended for use by pregnant or breastfeeding women.

When it comes to preventing or eliminating the formation of estrogens especially after the end of a steroid cycle, Nolvadex or Tamoxifen Citrate is one of the most trusted of all antiestrogens.

Nolvadex or Tamoxifen Citrate is considered by many as the best antiestrogen in town as it can easily increase the serum levels of testosterone besides eliminating or reducing the formation of “harmful” estrogens, especially after the end of a steroid cycle. This antiestrogen is also used for improving the levels of luteinizing hormone and Follicle-stimulating hormone. The antiestrogen is also used to treat breast cancer and promoting effective functioning of both HDL and LDL lipid profiles.

The fact that Nolvadex only eliminates the “harmful” estrogens and not all estrogens (some estrogens are good for building muscles and normal body functioning) is something unique to this antiestrogen. This antiestrogen is admired by professional sportsmen such as bodybuilders and strength athletes making use of harsh or aromatizable steroids, which lead to estrogenic side effects such as gynecomastia and fluid retention that can be effectively treated with an antiestrogen as potent as Nolvadex.

The recommended dose of Nolvadex is 20-40 mg per day for beginners and 35-50 mg per day for experienced steroid users. The active ingredient in Nolvadex tablets is tamoxifen citrate and its inactive ingredients are carboxymethylcellulose calcium, magnesium stearate, mannitol, and starch.

When of a low grade or abused, use of Nolvadex can lead to side effects such as hot flashes, depression, dizziness, headache, and vaginal dryness.

When it comes to inhibiting the formation of estrogens during or after a steroid cycle, Femara is a trustworthy antiestrogen. Read on!

Femara, which is also known as Letrozole, is considered to be an exceptional drug for treating infertility and inhibiting estrogen formation.

Having an approximate active life of 2-4 days, Femara belongs to the category of oral aromatase inhibitors. Femara allows users to raise the levels of luteinizing hormone, follicle-stimulating hormone, and sex hormone-binding globulin to a considerable extent. In addition to that, this preferred antiestrogen is good enough to be a part of every bulking or cutting cycle.

In addition to this, Femara is also useful for reducing the potential risks of acne and gynecomastia. Femara blocks the enzyme aromatase that blocks estrogen production to a significant extent. The results after using Femara can be dramatic, to say the least. Use of Femara also leads to improved muscle quality without holding excess water.

In the world of medicines, Femara is used to treat breast cancer after failure of traditional therapies such as Tamoxifen therapy.

Recommended Dose

The recommended dose of Femara is 0.5-2.5 mg per day, with or without meals.

Possible Side effects

When abused or of a low-grade quality, Femara can lead to possible side effects such as acne, liver toxicity, hair thinning, and hot flushes.

Storage Conditions

Femara tablets need to be kept at a controlled room temperature of 25°C (77°F) with excursions permitted up to 15-30°C (59-86°F). The tablets must be kept at a good distance away from pets, children, direct sunlight, moisture, and unauthorized usage.

When it comes to an effective aromatase inhibitor, the mention of Cytadren comes at the first place.

Cytadren, which is also known as Aminoglutethimide, is an effective inhibitor of desmolase (an enzyme required for steroid production in the body). This drug is considered to be exemplary when use of aromatizable steroids is the basic intention of steroid users.

In the world of bodybuilding, Cytadren is an effective antiestrogen especially in the stage of post cycle therapy. Since this drug can easily inhibit the conversion of cholesterol to pregnenolone, it is admired by bodybuilders when it comes to reducing or eliminating the formation of estrogens.

It is considered to be second to none while a sportsman or bodybuilder is dieting for a contest. The characteristics of this drug are of great worth when the circulating androgens get totally replaced by synthetic androgens during dieting and before the contest. This is an effective antiestrogen for all those sportsmen who want to stay away from the possible side effects of harsh steroids or aromatizable steroids that could have led to side effects such as gynecomastia and fluid retention.

In addition to all these benefits, Cytadren is also useful because of its unique anti-depressive properties.

Recommended Dose

The recommended dose of Cytadren is 100-200 mg/day, with or without meals. The use of Cytadren must be recommended by a qualified medical practitioner else a situation of substance abuse is not far away.

We hope that this information on Cytadren, the effective aromatase inhibitor, helped you to gain a clear and complete insight on this miracle drug.

When it comes to optimizing benefits of anabolic steroids at the end of a steroid cycle, Clomid is one name that is admired by one and all.

Clomid, which is also known as Clomiphene Citrate, is an effective antiestrogen when it comes to improving recovery of body’s natural testosterone production after a steroid cycle. In addition to that, Clomid is also admired for minimizing the potential risk of gynecomastia during a cycle employing aromatizable steroids.

In addition to these benefits, Clomid is useful for improving the level of blood cholesterol and acting as an effective agonist in bone tissue besides minimizing the adverse effect of exercise-induced damage of muscle tissue.

This orally administered, nonsteroidal, ovulatory stimulant has the chemical name of 2-[p-(2-chloro-1,2-diphenylvinyl)phenoxy] triethylamine citrate (1:1). Its molecular weight is 598.09 g/mol at the base and its molecular formula is C₂₆H₂₈ClNO • C₆H₈O₇.

The active ingredient of Clomid tablets is 50 mg clomiphene citrate USP and its inactive ingredients include corn starch, lactose, magnesium stearate, pregelatinized cornstarch, and sucrose.

Recommended Dose

The recommended dose of Clomid is 50 mg/day, with or without meals, for a period of five days at a stretch.

Possible Side Effects

When abused or a low-grade quality, Clomid can lead to possible side effects such as blurred vision, lights, floaters, waves, headache, vomiting, nausea, and depression.

Clomid tablets are required to be kept at a controlled room temperature 59-86°F (15-30°C).

We hope that this information on Clomid, the effective antiestrogen, was helpful to you in more than just a way.

In the worlds of performance enhancing drugs, antiestrogens, and steroids, Arimidex is one name that is trusted by one and all especially when steroid cycles involve harsh or aromatizable steroids.

Arimidex, also known as Anastrozole or Liquidex, was initially developed as a drug to treat advanced breast cancer in women. But it slowly gained popularity as a new class of third-generation selective oral aromatase inhibitor. This wonder drug is effective for inhibiting the enzyme aromatase besides inhibiting the production of estrogens, especially after use of harsh or aromatizable drugs during steroid cycles.

It is worth noting here that Arimidex is better than Nolvadex, another antiestrogen, because Arimidex is able to provide improved and dramatic results when compared to Nolvadex.

Even at low doses of 0.25-1.0 mg per day, Arimidex is an exceptional antiestrogen that can inhibit potential risks such as fluid retention and gynecomastia to a great extent. This also means that muscle quality is greater and without any side effects with Arimidex. This oral aromatase inhibitor has an active life of approximately 42-48 hours and can reduce the level of blood pressure when coupled with aromatizable steroids during a steroid cycle.

It is important to note that use of Arimidex should be initiated only after a medical recommendation so that existing allergies to ingredients of Arimidex and possible side effects can be completely ruled out. If this is not taken care of, Arimidex abuse can lead to side effects such as bone pain, peripheral edema, dyspnea, hot flashes, arthritis, insomnia, depression, nausea, and vomiting.